Skip to main content
Top

2023 | OriginalPaper | Chapter

3. Discovery of Small-Molecule Modulators of Protein–RNA Interactions by Fluorescence Intensity-Based Binding Assay

Author : Dr. Wan Gi Byun

Published in: Discovery of Small-Molecule Modulators of Protein–RNA Interactions for Treating Cancer and COVID-19

Publisher: Springer Nature Singapore

Activate our intelligent search to find suitable subject content or patents.

search-config
loading …

Abstract

Protein–RNA interactions (PRIs) play crucial roles in the regulation of various key steps in gene expression.

Dont have a licence yet? Then find out more about our products and how to get one now:

Springer Professional "Wirtschaft+Technik"

Online-Abonnement

Mit Springer Professional "Wirtschaft+Technik" erhalten Sie Zugriff auf:

  • über 102.000 Bücher
  • über 537 Zeitschriften

aus folgenden Fachgebieten:

  • Automobil + Motoren
  • Bauwesen + Immobilien
  • Business IT + Informatik
  • Elektrotechnik + Elektronik
  • Energie + Nachhaltigkeit
  • Finance + Banking
  • Management + Führung
  • Marketing + Vertrieb
  • Maschinenbau + Werkstoffe
  • Versicherung + Risiko

Jetzt Wissensvorsprung sichern!

Springer Professional "Technik"

Online-Abonnement

Mit Springer Professional "Technik" erhalten Sie Zugriff auf:

  • über 67.000 Bücher
  • über 390 Zeitschriften

aus folgenden Fachgebieten:

  • Automobil + Motoren
  • Bauwesen + Immobilien
  • Business IT + Informatik
  • Elektrotechnik + Elektronik
  • Energie + Nachhaltigkeit
  • Maschinenbau + Werkstoffe




 

Jetzt Wissensvorsprung sichern!

Literature
1.
go back to reference Re A, Joshi T, Kulberkyte E, Morris Q, Workman CT (2014) Methods Mol Biol 1097:491–521CrossRef Re A, Joshi T, Kulberkyte E, Morris Q, Workman CT (2014) Methods Mol Biol 1097:491–521CrossRef
2.
go back to reference Lukong KE, Chang K-W, Khandjian EW, Richard S (2008) Trends Genet 24:416–425; Conlon EG, Manley JL (2017) Genes Dev 31:1509–1528 Lukong KE, Chang K-W, Khandjian EW, Richard S (2008) Trends Genet 24:416–425; Conlon EG, Manley JL (2017) Genes Dev 31:1509–1528
3.
go back to reference Hentze MW, Castello A, Schwarzl T, Preiss T (2018) Nat Rev Mol Cell Biol 19:327–341CrossRef Hentze MW, Castello A, Schwarzl T, Preiss T (2018) Nat Rev Mol Cell Biol 19:327–341CrossRef
4.
go back to reference Ellis JJ, Broom M, Jones S (2007) Proteins Struct Funct Bioinf 66:903–911CrossRef Ellis JJ, Broom M, Jones S (2007) Proteins Struct Funct Bioinf 66:903–911CrossRef
5.
go back to reference Nasti R, Rossi D, Amadio M, Pascale A, Unver MY, Hirsch AKH, Collina S (2017) J Med Chem 60:8257–8267; Maurer CK, Fruth M, Empting M, Avrutina O, Hoßmann J, Nadmid S, Gorges J, Herrmann J, Kazmaier U, Dersch P, Meller R, Hartmann RW (2016) Future Med Chem 8:931–947; Lim D, Byun WG, Koo JY, Park H, Park SB (2016) J Am Chem Soc 138:13630–13638; Lorenz DA, Kaur T, Kerk SA, Gallagher EE, Sandoval J, Garner AL (2018) ACS Med Chem Lett 9:517–521; Wang L, Rowe RG, Jaimes A, Yu C, Nam Y, Pearson DS, Zhang J, Xie X, Marion W, Heffron GJ, Daley GQ, Sliz P (2018) Cell Rep 23:3091–3101; Rzuczek SG, Colgan LA, Nakai Y, Cameron MD, Furling D, Yasuda R, Disney MD (2017) Nat Chem Biol 13:188–193 Nasti R, Rossi D, Amadio M, Pascale A, Unver MY, Hirsch AKH, Collina S (2017) J Med Chem 60:8257–8267; Maurer CK, Fruth M, Empting M, Avrutina O, Hoßmann J, Nadmid S, Gorges J, Herrmann J, Kazmaier U, Dersch P, Meller R, Hartmann RW (2016) Future Med Chem 8:931–947; Lim D, Byun WG, Koo JY, Park H, Park SB (2016) J Am Chem Soc 138:13630–13638; Lorenz DA, Kaur T, Kerk SA, Gallagher EE, Sandoval J, Garner AL (2018) ACS Med Chem Lett 9:517–521; Wang L, Rowe RG, Jaimes A, Yu C, Nam Y, Pearson DS, Zhang J, Xie X, Marion W, Heffron GJ, Daley GQ, Sliz P (2018) Cell Rep 23:3091–3101; Rzuczek SG, Colgan LA, Nakai Y, Cameron MD, Furling D, Yasuda R, Disney MD (2017) Nat Chem Biol 13:188–193
7.
8.
10.
go back to reference D’Agostino VG, Sighel D, Zucal C, Bonomo I, Micaelli M, Lolli G, Provenzani A, Quattrone A, Adami V (2019) SLAS Discovery 24:314–331CrossRef D’Agostino VG, Sighel D, Zucal C, Bonomo I, Micaelli M, Lolli G, Provenzani A, Quattrone A, Adami V (2019) SLAS Discovery 24:314–331CrossRef
12.
15.
go back to reference Sampson VB, Rong NH, Han J, Yang Q, Aris V, Soteropoulos P, Petrelli NJ, Dunn SP, Krueger LJ (2007) Cancer Res 67:9762–9770CrossRef Sampson VB, Rong NH, Han J, Yang Q, Aris V, Soteropoulos P, Petrelli NJ, Dunn SP, Krueger LJ (2007) Cancer Res 67:9762–9770CrossRef
16.
go back to reference Johnson SM, Grosshans H, Shingara J, Byrom M, Jarvis R, Cheng A, Labourier E, Reinert KL, Brown D, Slack FJ (2005) Cell 120:635–647CrossRef Johnson SM, Grosshans H, Shingara J, Byrom M, Jarvis R, Cheng A, Labourier E, Reinert KL, Brown D, Slack FJ (2005) Cell 120:635–647CrossRef
18.
go back to reference Piskounova E, Polytarchou C, Thornton JE, LaPierre RJ, Pothoulakis C, Hagan JP, Iliopoulos D, Gregory RI (2011) Cell 147:1066–1079CrossRef Piskounova E, Polytarchou C, Thornton JE, LaPierre RJ, Pothoulakis C, Hagan JP, Iliopoulos D, Gregory RI (2011) Cell 147:1066–1079CrossRef
19.
go back to reference Unruh JR, Gokulrangan G, Wilson GS, Johnson CK (2005) Photochem Photobiol 81:682–690CrossRef Unruh JR, Gokulrangan G, Wilson GS, Johnson CK (2005) Photochem Photobiol 81:682–690CrossRef
21.
go back to reference Liu Y, Miao K, Dunham NP, Liu H, Fares M, Boal AK, Li X, Zhang X (2017) Biochemistry 56:1585–1595CrossRef Liu Y, Miao K, Dunham NP, Liu H, Fares M, Boal AK, Li X, Zhang X (2017) Biochemistry 56:1585–1595CrossRef
22.
go back to reference Nowak JS, Choudhury NR, de Lima Alves F, Rappsilber J, Michlewski G (2014) Nat Commun 5:3687ADSCrossRef Nowak JS, Choudhury NR, de Lima Alves F, Rappsilber J, Michlewski G (2014) Nat Commun 5:3687ADSCrossRef
23.
go back to reference Lukinavičius G, Umezawa K, Olivier N, Honigmann A, Yang G, Plass T, Mueller V, Reymond L, Corrêa IR, Luo Z-G, Schultz C, Lemke EA, Heppenstall P, Eggeling C, Manley S, Johnsson K (2013) Nat Chem 5:132–139CrossRef Lukinavičius G, Umezawa K, Olivier N, Honigmann A, Yang G, Plass T, Mueller V, Reymond L, Corrêa IR, Luo Z-G, Schultz C, Lemke EA, Heppenstall P, Eggeling C, Manley S, Johnsson K (2013) Nat Chem 5:132–139CrossRef
24.
25.
go back to reference Lightfoot HL, Miska EA, Balasubramanian S (2016) Org Biomol Chem 14:10208–10216CrossRef Lightfoot HL, Miska EA, Balasubramanian S (2016) Org Biomol Chem 14:10208–10216CrossRef
27.
go back to reference Williams LK, Zhang X, Caner S, Tysoe C, Nguyen NT, Wicki J, Williams DE, Coleman J, McNeill JH, Yuen V, Andersen RJ, Withers SG, Brayer G (2015) D. Nat Chem Biol 11:691–696CrossRef Williams LK, Zhang X, Caner S, Tysoe C, Nguyen NT, Wicki J, Williams DE, Coleman J, McNeill JH, Yuen V, Andersen RJ, Withers SG, Brayer G (2015) D. Nat Chem Biol 11:691–696CrossRef
28.
29.
go back to reference Dias TA, Duarte CL, Lima CF, Proenca MF, Pereira-Wilson C (2013) Eur J Med Chem 65:500–510CrossRef Dias TA, Duarte CL, Lima CF, Proenca MF, Pereira-Wilson C (2013) Eur J Med Chem 65:500–510CrossRef
30.
go back to reference Verma AK, Singh H, Satyanarayana M, Srivastava SP, Tiwari P, Singh AB, Dwivedi AK, Singh SK, Srivastava M, Nath C, Raghubir R, Srivastava AK, Pratap R (2012) J Med Chem 55:4551–4567CrossRef Verma AK, Singh H, Satyanarayana M, Srivastava SP, Tiwari P, Singh AB, Dwivedi AK, Singh SK, Srivastava M, Nath C, Raghubir R, Srivastava AK, Pratap R (2012) J Med Chem 55:4551–4567CrossRef
32.
go back to reference Schlundt A, Heinz GA, Janowski R, Geerlof A, Stehle R, Heissmeyer V, Niessing D, Sattler M (2014) Nat Struct Mol Biol 21:671–678CrossRef Schlundt A, Heinz GA, Janowski R, Geerlof A, Stehle R, Heissmeyer V, Niessing D, Sattler M (2014) Nat Struct Mol Biol 21:671–678CrossRef
33.
go back to reference Leppek K, Schott J, Reitter S, Poetz F, Hammond MC, Stoecklin G (2013) Cell 153:869–881CrossRef Leppek K, Schott J, Reitter S, Poetz F, Hammond MC, Stoecklin G (2013) Cell 153:869–881CrossRef
35.
36.
go back to reference Bouktaib M, Lebrun S, Atmani A, Rolando C (2002) Tetrahedron 58:10001–10009CrossRef Bouktaib M, Lebrun S, Atmani A, Rolando C (2002) Tetrahedron 58:10001–10009CrossRef
37.
go back to reference Thapa M, Kim Y, Desper J, Chang K-O, Hua DH (2012) Bioorg Med Chem Lett 22:353–356CrossRef Thapa M, Kim Y, Desper J, Chang K-O, Hua DH (2012) Bioorg Med Chem Lett 22:353–356CrossRef
Metadata
Title
Discovery of Small-Molecule Modulators of Protein–RNA Interactions by Fluorescence Intensity-Based Binding Assay
Author
Dr. Wan Gi Byun
Copyright Year
2023
Publisher
Springer Nature Singapore
DOI
https://doi.org/10.1007/978-981-19-7814-2_3